Medicinal Chemistry

6^th World Congress on Medicinal Chemistry and Drug Design

June 07-08, 2017 Milan, Italy

Posters & Accepted Abstracts

• 5α-steroidal amines: Synthesis and biological activity

  N Nadaraia, M Merlani, N Barbakadze, N Amiranashvili and M Kakhabrishvili

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• Successful strategies for recruitment of african americans into clinical studies

  Jane Otado

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• Synthesis of oseltamivir using Diels-Alder reaction of 1, 3-butadiene bearing 2-carboxy and 4-alkoxy substituents

  Szu-Han Chen

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• Design and synthesis of sugar phosphates for inhibition of tuberculosis maltosyl transferase

  Wei-Hsin Hsu

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• Mapping the vibrational transition-state conformational change in enzymes for drug design

  Yun Lu

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• Morphological and structural features of adenovirus particles by reacting with bacterial cell

  Anna Golovan, S I Voychuk, I L Garmasheva, O Yu Povnitsa, L B Bilyavska, O N Vasilyuk, K S Naumenko and Yu B Pankivska

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• Early findings in the development of an enzymatically triggered nanoformulation

  Daniel Ehrsam, Fabiola Porta, Mouhssin Oufir, Dominik Witzigmann, Jorg Huwyler, Matthias Hamburger and Henriette E Meyer zu Schwabedissen

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• Pyrroles - A novel synthetic method for pyrrole derivatives from nitrodienes

  Mohamed A El-Atawy, F Ferretti and F Ragaini

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• Apoptotic mechanism of compounds with antiproliferative activity from Bursera microphylla resin

  Francisco H. González-Gutierrez; Luisa A. Rascon-Valenzuela, Olivia Valenzuela-Antelo, M.C. Marcotullio and Ramon E. Robles-Zepeda

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• New 1, 2, 5-oxadiazole Pt(II)complex endowed with STAT3 inhibitory properties as promising anticancer agent

  Arianna Gelain, Stefania Villa, Fiorella Meneghetti, Federica Porta, Giorgio Facchetti, Nicola Ferri, Akira Asai3, Valentina Gandin, Cristina Marzano and Isabella Rimoldi

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• Synthesis of novel furan-based antituberculars potentially targeting the methionine aminopeptidases (MtMetAP1a)

  Arianna Gelain, Stefania Villa, Matteo Mori, Laurent R Chiarelli, Luca Costantino, Tiziano Tuccinardi and Fiorella Meneghetti

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• Study of protector effect of chemlal olive leaves extract on nephropathy induced by mercury in mouse

  Dekdouk Nadia, Ameddah Souad, Menad Ahmed, De Tommasi Nunziatina, Malafronte Nicola and Mekkio Ratiba

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• Why the drug solutions may cause inflammation at the injection site

  Kasatkin A and Urakov A

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• The role of technologies of nonlinear stimulation in the treatment of brain diseases and potential of their applications in healthy individuals

  Marina V Zueva

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• The study in vitro of the effects of the inhalant corticosteroids on oral and laryngeal mucosa

  Didier Alexandre, Menicagli Roberto and Marotta Ortensio

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• Drug hunting vs. drug fishing

  Youssef L Bennani

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• Adapting DNA-encoded library technology for fragment-based drug discovery

  Mike Thompson

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• Phenotypes of a novel series of 3-phosphoglycerate dehydrogenase inhibitors

  Nello Mainolfi

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• Synthesis and anticancer activity of 6-aryl-2-naphthyl-imidazo[2,1 b][1,3,4]thiadiazole

  Subhas S Karki, Chudamani B, Sujeet Kumar, Hiroshi Sakagami, Yoshiko Masuda, Satoshi Yokose, Yoshihiro Uesawa, Hajime Kagaya, Erik De Clercq and Dominique Schols

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• Comparison of heavy metal levels in the fish oil obtained from the janitor fish (Pterygoplichthys disjunctivus) from Marikina River and Laguna de Bay using atomic absorption spectrometry

  A R Lapuz, Guan A N, Ambay R V and Mendoza J D

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• Investigation of effect of medium on volumetric and ultrasonic studies of pharmaceutical excipients

  Bushra Naseem

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• The great potential of phenolic compounds isolated from Limonium densiflorum to quench and protect human cell against free radicals

  Faten Medini, Manel oueslati, Jean Legault and Riadh Ksouri

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• Cyclopentenes for anti-tuberculosis and antibiotics

  Hadia Almahli and Stephen P Fletcher

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• Synthesis and neuroprotective activity of novel 5,6-diaryl-1,2,4-triazine derivatives with ethyl acetate moiety against H2O2 and Aβ-induced neurotoxicity

  Hamid Irannejad and Tuba Tuylu Kucukkilinc

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• Anticancer activity of some [1,2,4]triazepino[2,3-a] quinazoline derivatives: Monolayer and multicellular spheroids in vitro models

  Hanem M Awad

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• In the pursuit of ideal hits for antifungal research

  Jeanmart Stephane

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• Structure-based design of subtype selective antagonists for the ionotropic glutamate receptors: Successes and failures

  Lennart Bunch

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• Protective effect of the standardized extract of Holmskioldia sanguinea on tumor bearing mice

  Mahesh Pal, Tripti Mishra, Ch V Rao and D K Upreti

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• Novel 5-susituated analogues of 4H-3-(2-phenoxy)phenyl–1,2,4-triazole derivatives as agonists of benzodiazepine receptors with anxiolytic effect

  Mehrdad Faizi, Aliasghar Peyvandi and Sayyed Abbas Tabatabai

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• Quadruplex DNA stabilizing agents as potential anti-cancer therapeutics

  Mrinalkanti Kundu

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• Isoconversional approach for non-isothermal decomposition of un-irradiated and photon-irradiated 5-fluorouracil

  Refaat M Mahfouz, Hala Sh Mohamed and Abdel Rahman A Dahy

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• Passiflora incarnata L. of endophytic fungi rooted flavone chrysin (5,7-dihydroxy flavone) and gold nanoparticles towards anticancer activity

  Sivaperumal Sivaramakrishnan

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• The study on serum protein spectrum expression changes for patients with gastrointestinal disease before and after acupuncture

  Yanhong Gao

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• Design and development of ureas and amides as p38 kinase inhibitors

  Ravindra Kulkarni, Achaiah Garlapati, Stefan Laufer and Chandrashekhar V M

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