Medicinal Chemistry

2^nd International Conference on PHARMACEUTICAL CHEMISTRY

October 02-04, 2017 Barcelona, Spain

Posters & Accepted Abstracts

• Nitroxide-modified chitosans with enhanced antioxidant potential

  Vasily Sen, Nikolai Neshev, Anastasiya Balakina, Viktoriya Mumyatova, Alexei Terentiev and Evgeny Pliss

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• N-aryl effects on the catalyst reactivity of imidazolylidene in a3→d3-umpolung addition: Structural study and mechanistic investigation

  Tetsuo Narumi, Ryuji Kyan, Kohei Sato and Nobuyuki Mase

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• Analysis of the polar solvents influence on the mechanism of the inhibited oxidation of unsaturated compounds

  Sergey Lednev and Andrey Sirik

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• Influence of solvation on the mechanism of the hydroperoxide radicals' addition to the π-bonds of trans 1,2-and 1,4-diphenylbutadiyne-1,3

  Roman Pliss, Mikhail Soloviev, Evgeny Pliss, Aleksey Grobov and Andrey Sirik

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• Mathematical modelling of polychromatic light photokinetics

  Mohammed Alqarni and Mounir Maafi

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• High-throughput screening to identify novel inhibitors of human α-methylacyl-CoA racemase 1A (AMACR; P504S)

  Matthew D Lloyd, Yoana D Petrova, Hannah Matan, Louise Chow, Angel Wai, Kairavi Raja, Maksims Yevglevskis, Amit Nathubhai, Guat L Lee, Tony D James, Michael D Threadgill and Timothy J Woodman

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• The secrets and potential of a novel cyclic antimicrobial and cell penetrating peptide

  Margitta Dathe, Kathi Scheinpflug, Christof Junkes, Mojtaba Bagheri, Henrik Strahl and Oxana Krylova

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• Nitroxyl radicals as antioxidants against lipid peroxidation: An in vitro study

  Ivan Tikhonov and Leonid Borodin

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• Oxidative stress simulation by radical-chain oxidation of vinyl compounds

  Evgeny Pliss, Mikhail Soloviev, Aleksey Grobov, Roman Pliss and Andrey Sirik

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• A novel one pot two-step strategy for regio-chemoselective synthesis of new 3-methyl6-arylpyridazine4-carboxamides and 5-oxo-3-aryl-5,6-dihydropyrido[4,3-c]pyridazine-8-carbaldehydes

  Ali Aghaye Lotf va Ata, Mehdi Rimaz and Mohammad Mehdi Baradarani

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• Synthesis of some novel 2-(substituted thio)-N-(5-methyl-4-phenylthiazol-2-yl)acetamide and anticancer activity evaluation

  Asaf Evrim Evren, Leyla Yurttas, Busra Ekselli and Gulsen Akalin-Ciftci

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• Synthesis of some novel N-(6-substituted benzothiazole-2-yl)-2-(4-substituted piperazin-1-yl) asetamide derivatives and evaluation their anticancer activity

  Büsra Ekselli, Gülsen Akalın-Ciftci, Asaf Evrim Evren And Leyla Yurttas

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• Conjugated nitroalkenes in reactions with azomethine imines: Synthesis of tetrahydropyrazolo[1,2-a] pyrazolone derivatives

  Nikolay S. Zimnitskiy, Vladislav Yu. Korotaev, Igor B. Kutyashev, Alexey Yu. Barkov and Vyacheslav Ya. Sosnovskikh

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• An optimized process for supercritical CO2 extraction of high-value components from Artemisia annua L for cosmetic applications

  Rosana M. Alberici Oliveira

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• Fingernails: Development and validation of a rapid and sensitive method for quantification of cocainics by LC-ESI-MS/MS

  Nascimento H, Loss C. G. ; Santos Jr J C, Jara J L P, Borgo, A P, Filho, P C M, Guidugli R B F, Eberlin M N and Höehr N F

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• Rapid and sensitive method for simultaneous determination of first-line anti-tuberculosis drugs in human plasma by HPLC-MS/MS: Application to therapeutic drug monitoring

  Shouhong GAO and Wansheng CHEN

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• Homology modelling of different leishmanolysin (gp63) from leishmania spp. and molecular docking of flavonoids

  Jairo Mercado-Camargo, Leonor Cervantes-Ceballos and Harold Gómez-Estrada

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• An In silico approach to discovering inhibitiors of trypanothione reductase from leishmania (viannia) panamensis.

  Leonor Cervantes-Ceballos; Elkin Torres Sierra; María Luisa Serrano García and Harold Gómez-Estrada

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• In vitro evaluation of cytotoxicity and leishmanicidal activity of terpens isolated from the leaves of malachra alceifolia

  Harold Gómez-Estrada, Leonor Cervantes-Ceballos and Sara Robledo-Restrepo

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• Cascade approach to modification of lactone macrolide antibiotics

  Krystian Pyta, Katarzyna Pyta-Klich, Anna Janas, Joanna Domagalska and Piotr Przybylski

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• Sizing α, β and γ cyclodextrins by capillary electrophoresis and indirect UV detection

  Yin Zhou

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• Novel quinazoline derivative as RAF Inhibitor

  Shih-Chieh Yen, Chu-Bin Liao, Hung-Jyun Huang, Ju-Ying Yang, Yen-Hsi Liu, Sian-Yi Ciou, Mann-Yan Kuo, and Shao-Zheng Peng

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• Determination of heavy metal(PB) content in mineral water produced in IRAN by Flameless Atomic Absorption Spectroscopy (FAAS)

  Rasoul Kazemi, Orkideh gorban dadras and Masoud amanlou

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• Synthesis of novel spiro dipyrazolo[3,4-b: 4΄,3΄-e]pyridine

  Bahman Ebrahimi Saatluo and Mehdi M Baradarani

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• DBU/H2O as an efficient, eco-friendly and inexpensive catalyst for transesterification and transacylation reactions

  Elaheh Akbarzadeh and Elham Pour Namdari

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• AB initio and DFT study of energetic, stability, and nuclear magnetic resonance of BN nanotube

  Elham Pournamdari and Elaheh Akbarzadeh

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• In vitro antiproliferative, antioxidant, and apoptosis-inducing activities of dried flower buds of clove extract on human gastric carcinoma

  Ali Karimi and Mohammad-taghi Moradi

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• Synthesis and cytotoxic properties of new derivatives of dicarboximides

  M Napiorkowska, M Cieelak, K Krolewska, J Kazmierczak-Baranska and B Nawrot

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• Discovery of novel aryl hydrocarbon receptor (AhR) antagonists using homology modelling and ligand-based drug design

  Carlos Henrique Tomich de Paula da Silva, Larissa Pernomian and Joao Gabriel Curtolo Poiani

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• Structural aspects of PtP2CNL and PtP2CBL derivatives of organophosphines in organoplatinum complexes

  Peter Mikus and Milan Melnik

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• Synthesis and biological investigation of phosphabetaine derivatives

  I Galkina, D Bakhtiyarov, Y Bakhtiyarova, M Shulaeva, O Pozdeev, S Egorova and V Galkin

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• A combinatorial methodology for the discovery of new agents with insect repellent properties

  Eftychia Kritsi, Spyros Zografos, and Panagiotis Zoumpoulakis

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• New Systems for Organocatalytic Asymmetric Epoxidation

  Philip C Bulman Page

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• Synthesis and Structures of Pincer-Type Rhodium(III) complexes; Reactivity Toward Small Biomolecules, calf thymus DNA (CT-DNA) and bovine serum albumin (BSA)

  Jovana V Bogojeski, Milan M Milutinovi,ad,Olivera Klisuric, Sofi K C Elmroth, Andreas Scheurer and Zivadin D Bugarcic

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• Novel Potential Antihyperlipidaemic Agents Derived From Heterocyclic-2-carboxamides

  Yusuf M. Al-Hiari

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• Trysts with Anti-Cancer Drug Designing - Design Synthesis and Evaluation Some Chromone and β-Ionone Based Anticancer Molecules

  Mohan Paul Singh Ishar

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• Caffeic Acid-Derived Biopolyether from Medicinal Plants as Anticancer Agent

  Vakhtang Barbakadze

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• Dynamic combinatorial approch as synthetic strategy for the formation of non-viral vectors for gene therapy

  Lilia Clima

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• Unusual Reaction of Phenylation and New Appoach for the Synthesis of Tritium Labeled Biomarkers with Quaternary Heterocyclic Nitrogen Atom

  Nadezhda Shchepina

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• Synthesis of heteroaryl-substituted pyrazolo[1,5-a]pyrimidines by recyclization of pyrimidinium salts

  Gevorg G. Danagulyan

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• Newly potent opioid peptides with analgesic activity containing a xylene bridge

  Adriano Mollica

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• Diverse and versatile synthesis of bioactive heterocyclic compounds from keto acids

  Ahmed Majeed Hsskia

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• Design and synthesis of inhibitors of the GDP-Mannose Pyrophosphorylase(GDP-MP)

  Christian Cave

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• Development of inhibitors of the cysteine proteases rhodesain of T. b. rhodesiense and falcipain-2 of P. falciparum

  Roberta Ettari

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• Nano anti-cancer drugs: Hope for future

  Imran Ali

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• New synthetic methods for medicinal chemistry

  Markus R. Heinrich

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• Transition metal complexes/organometallic compounds as anticancer/anti HIV drugs or in pharmaceutical industry

  Prakash Kinthada

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• Designed peptidomimetics disrupt protein-protein interactions mediating amyloid protein aggregation

  Sandrine Ongeri

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• A Modern In Vivo PK Paradigm: Combining Snapshot, Rapid and Full PK Approaches to Support Early Drug Discovery

  Tove Tuntland

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• Arylglyoxals as precursors for synthesis of N-hydroxyhydantoins, N-alkoxyhydantoins and thiohydantoins in mild conditions

  Victor Shtamburg

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• Designing antitubercular agents exploring Mycobactin biosynthetic patway

  Venkatesan Jayaprakash

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• New drug development and problem-solving in the pharmaceutical industry

  Satinder Ahuja

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• Selective Electrochemical Oxidation for Chemical Synthesis and Fuel Generation

  Stafford W. Sheehan

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