Medicinal Chemistry

6^th World Congress on Medicinal Chemistry and Drug Design

June 07-08, 2017 Milan, Italy

Scientific Tracks Abstracts

• Quantification of some medical preparations of the plant origin

  Malkhaz Getia, Vakhtang Mshvildadze, Zurab Kemoklidze, Nana Gorgaslidze, Andre Pichette and Genri Dekanosidze

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• Phospholipid-based prodrugs for the treatment of IBD: Drug targeting strategy

  Shimon Ben-Shabat, Arik Dahan, Ellen M Zimmerman and Aaron Aponick

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• Drug design via a scaffold hopping strategy: Case studies on discovery of clinical candidates H3 receptor antagonist and β-tryptase inhibitor

  Zhongli Gao

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• Drug design via a scaffold hopping strategy: Case studies on discovery of clinical candidates H3 receptor antagonist and β-tryptase inhibitor

  Zhongli Gao

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• Nutraceuticals in gastrointestinal ailments: An emerging paradigm

  Matteo Micucci, Alberto Chiarini, Monica Cevenini, Rita Aldini and Roberta Budriesi

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• Pathogenesis of alimentary diabetes: recovery by loss of 20% body weight, and by attainment of initial hunger as well as of low BG before meals

  Gaia Cecchia

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• The new steroids from Silene montbretiana

  Hilal Kilinc, Milena Masullo, Tamer Karayildirim, Sonia Piacente and Ozgen Alankus

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• Therapeutic important medicinal plants and way forward

  Neeraj Tandon

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• Continuous bio manufacturing of extracellular vesicles

  William G Whitford and Alexander Aristarkhov

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• α,β-unsaturated compounds derived from arylamines as possible new treatment against leukemia

  Sanchez-Labastida Luis Angel, Bribiesca-Carlos Jose, Andrade-Jorge Erik, Vasquez-Moctezuma Ismael and Trujillo-Ferrara Jose Guadalupe

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• α,β-unsaturated compounds derived from arylamines as possible new treatment against leukemia

  Sanchez-Labastida Luis Angel, Bribiesca-Carlos Jose, Andrade-Jorge Erik, Vasquez-Moctezuma Ismael and Trujillo-Ferrara Jose Guadalupe

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• Development of analytical procedure for the standardization of bromelain from the pineapple (Ananas comosus (L.) Merr.)

  Nana Gorgaslidze, Nino Nizharadze, Liana Nadirashvili, George Erkomaishvili and Malkhaz Getia

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• CZ415, a highly selective mTOR inhibitor showing in vivo efficacy in a collagen induced arthritis (CIA) model

  Giovanna Bergamini

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• β-strand mimicry: Exploring oligothienylpyridine foldamers

  Jana Sopkova-de Oliveira Santos, Marie Jouanne, Anne Sophie Voisin-Chiret, Remi Legay, Sebastien Coufourier and Sylvain Rault

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• Bioactive natural products from Symphytum (Boraginaceae)

  L Amiranashvili, L Gogilashvili, M Merlani and V Barbakadze

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• In Vitro and In Silico Studies of Peptide Inhibitors of Antibiotic Resistance Enzymes

  Laleh Alisaraie, Blake Hollett Power, Nathan Smith and Brandon Downer

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• 5α-Steroidal hydrazones: Synthesis and biological activity

  Maia Merlani, Nana Nadaraia, Lela Amiranashvili, Mery Kakhabrishvili and Nana Barbakadze

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• Synthesis and characterization of 2-((4R,4aR,5aS,6S)-1,3-dioxo3m3a,4,4a,5,5a6,6a-octahydro-4,6- ethenocyclopropa[f]isoindol-2(1H)-yl)-N-(substituted phenyl) acetamides anticipated to have HIV- 1 activity

  Abdulmajeed S H AlSamarrai and Noor H Abdulla

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• Identification of thiadiazinyl-coumarin derivatives as dengue virus-2 NS2B/NS3 protease inhibitors

  Hasnah Osman, Mohd Zaheen Hassan and Nadirah Zawani Mohd Nesfu

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• Therapeutic effects of trehalose liposomes against carcinoma along with apoptosis in vitro and in vivo

  Yoko Matsumoto

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• Ganoderma lucidum-cytotoxic effects and cytokine gene induction as compared with the immunobladder® BCG in murine MB49 cells

  John W M Yuen, Cyrus K C Ho, Tony S S To and Chi-Fai Ng

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• Disabling essential enzyme motion for catalysis: An efficient approach for shikimate kinase inhibition

  Concepcion Gonzalez-Bello

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• Enzyme triggered nanomaterial for cancer therapy

  Fabiola Porta

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• A new class of β-lactam antibiotics active against drug-sensitive and drug-resistant Mycobacterium tuberculosis

  Monika I Konaklieva, Rostislav Kuskovsky, Kriti Arora, Helena I Boshoff and Clifton E Barry

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• Host DHFR-directed cycloguanil analogues endowed with promising activity against influenza virus and respiratory syncytial virus

  Michele Tonelli

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• Design of new drugs: Challenges for the rational development of novel ligands with affinity for G-proteincoupled receptors

  Jose R Bahena Herrera, Erik Andrade Jorge and Jose G Trujillo Ferrara

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